抄録
A synthetic approach to eudistomin via a β-lactam fused bicyclic oxathiazepin intermediate is described. A β-lactam fused oxathiazepin derivative was synthesized by intramolecular 7-membered oxime ether formation and subsequent face-selective reduction of the C-N double bond. A fully functionalized orthoalkenylphenylthioanilide bearing oxathiazepin ring was then prepared and construction of the indole skeleton under several radical-mediated conditions was examined.
| 本文言語 | English |
|---|---|
| ページ（範囲） | 738-740 |
| ページ数 | 3 |
| ジャーナル | Synlett |
| 号 | 5 |
| 出版ステータス | Published - 2003 5月 1 |
| 外部発表 | はい |
ASJC Scopus subject areas
- 有機化学