Solid-phase synthesis of indolecarboxylates using palladium-catalyzed reactions

Kazuo Yamazaki, Yosuke Nakamura, Yoshinori Kondo

研究成果: Article査読

103 被引用数 (Scopus)

抄録

Polymer-supported, palladium-catalyzed cyclization reactions effectively synthesized indolecarboxylates. Palladium-catalyzed carbon - carbon bond-forming reactions of immobilized enaminoesters followed by transesterification yielded indole 2- or 3-carboxylates with various functional groups on the benzene ring. Indolecarboxylates were efficiently cyclized via an intramolecular palladium-catalyzed amination reaction of immobilized N-substituted dehydrohalophenylalanines, and immobilized N-acetyl-dehydroalanines were efficiently converted into indolecarboxylates via tandem Heck-amination reactions.

本文言語English
ページ(範囲)6011-6019
ページ数9
ジャーナルJournal of Organic Chemistry
68
15
DOI
出版ステータスPublished - 2003 7 25

ASJC Scopus subject areas

  • 有機化学

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