Novel Methodology for the Efficient Synthesis of 3-Aryloxindoles: [1,2]-Phospha-Brook Rearrangement-Palladium-Catalyzed Cross-Coupling Sequence

研究成果: Article査読

9 被引用数 (Scopus)

抄録

A novel methodology for the efficient synthesis of 3-aryloxindoles from isatin derivatives was developed. The methodology involves the formation of an oxindole having a phosphate moiety at the C-3 position via the [1,2]-phospha-Brook rearrangement under Bronsted base catalysis followed by palladium-catalyzed cross-coupling with aryl boron reagents. The one-pot synthesis of 3-aryloxindoles from isatin derivatives is also described.

本文言語English
論文番号st-2016-u0165-l
ページ(範囲)1848-1853
ページ数6
ジャーナルSynlett
27
12
DOI
出版ステータスPublished - 2016 7 21

ASJC Scopus subject areas

  • 有機化学

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