Synthesis of Ethoxyethynylarenes by the Palladium-Catalyzed Reaction of Aryl Iodides with Ethoxy(trialkylstannyl)acetylenes

Takao Sakamoto; Akito Yasuhara; Yoshinori Kondo; Hiroshi Yamanaka

doi:10.1248/cpb.42.2032

Synthesis of Ethoxyethynylarenes by the Palladium-Catalyzed Reaction of Aryl Iodides with Ethoxy(trialkylstannyl)acetylenes

Takao Sakamoto, Akito Yasuhara, Yoshinori Kondo, Hiroshi Yamanaka

PHA - Molecular Pharmaceutical Science

Research output: Contribution to journal › Article › peer-review

22 Citations (Scopus)

Abstract

Palladium-catalyzed reaction of aryl and heteroaryl iodides with ethoxy(trialkylstannyl)acetylenes gave the ethoxyethynylarenes and -heteroarenes, which were easily transformed by hydration reaction into ethyl areneacetates and heteroareneacetates.

Original language	English
Pages (from-to)	2032-2035
Number of pages	4
Journal	Chemical and Pharmaceutical Bulletin
Volume	42
Issue number	10
DOIs	https://doi.org/10.1248/cpb.42.2032
Publication status	Published - 1994

Keywords

aryl iodide
ethoxy(trialkylstannyl)acetylene
ethoxyethynylarene
ethyl areneacetate
palladium-catalyzed reaction

ASJC Scopus subject areas

Chemistry(all)
Drug Discovery

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title = "Synthesis of Ethoxyethynylarenes by the Palladium-Catalyzed Reaction of Aryl Iodides with Ethoxy(trialkylstannyl)acetylenes",

abstract = "Palladium-catalyzed reaction of aryl and heteroaryl iodides with ethoxy(trialkylstannyl)acetylenes gave the ethoxyethynylarenes and -heteroarenes, which were easily transformed by hydration reaction into ethyl areneacetates and heteroareneacetates.",

keywords = "aryl iodide, ethoxy(trialkylstannyl)acetylene, ethoxyethynylarene, ethyl areneacetate, palladium-catalyzed reaction",

author = "Takao Sakamoto and Akito Yasuhara and Yoshinori Kondo and Hiroshi Yamanaka",

year = "1994",

doi = "10.1248/cpb.42.2032",

language = "English",

volume = "42",

pages = "2032--2035",

journal = "Chemical and Pharmaceutical Bulletin",

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T1 - Synthesis of Ethoxyethynylarenes by the Palladium-Catalyzed Reaction of Aryl Iodides with Ethoxy(trialkylstannyl)acetylenes

AU - Sakamoto, Takao

AU - Yasuhara, Akito

AU - Kondo, Yoshinori

AU - Yamanaka, Hiroshi

PY - 1994

Y1 - 1994

N2 - Palladium-catalyzed reaction of aryl and heteroaryl iodides with ethoxy(trialkylstannyl)acetylenes gave the ethoxyethynylarenes and -heteroarenes, which were easily transformed by hydration reaction into ethyl areneacetates and heteroareneacetates.

AB - Palladium-catalyzed reaction of aryl and heteroaryl iodides with ethoxy(trialkylstannyl)acetylenes gave the ethoxyethynylarenes and -heteroarenes, which were easily transformed by hydration reaction into ethyl areneacetates and heteroareneacetates.

KW - aryl iodide

KW - ethoxy(trialkylstannyl)acetylene

KW - ethoxyethynylarene

KW - ethyl areneacetate

KW - palladium-catalyzed reaction

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JO - Chemical and Pharmaceutical Bulletin

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