Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis

Kazuo Yamazaki; Yosuke Nakamura; Yoshinori Kondo

doi:10.1039/b206378f

Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis

Kazuo Yamazaki, Yosuke Nakamura, Yoshinori Kondo

PHA - Molecular Pharmaceutical Science

Research output: Contribution to journal › Article › peer-review

43 Citations (Scopus)

Abstract

Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.

Original language	English
Pages (from-to)	2137-2138
Number of pages	2
Journal	Journal of the Chemical Society. Perkin Transactions 1
Volume	2
Issue number	19
DOIs	https://doi.org/10.1039/b206378f
Publication status	Published - 2002 Jul 2

ASJC Scopus subject areas

Chemistry(all)

Access to Document

10.1039/b206378f

Cite this

@article{60781e5bd9b44fd9adfa0a6e5f681818,

title = "Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis",

abstract = "Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.",

author = "Kazuo Yamazaki and Yosuke Nakamura and Yoshinori Kondo",

year = "2002",

month = jul,

day = "2",

doi = "10.1039/b206378f",

language = "English",

volume = "2",

pages = "2137--2138",

journal = "Journal of the Chemical Society. Perkin Transactions 1",

issn = "1470-4358",

publisher = "Chemical Society",

number = "19",

}

TY - JOUR

T1 - Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis

AU - Yamazaki, Kazuo

AU - Nakamura, Yosuke

AU - Kondo, Yoshinori

PY - 2002/7/2

Y1 - 2002/7/2

N2 - Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.

AB - Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.

UR - http://www.scopus.com/inward/record.url?scp=0036026270&partnerID=8YFLogxK

UR - http://www.scopus.com/inward/citedby.url?scp=0036026270&partnerID=8YFLogxK

U2 - 10.1039/b206378f

DO - 10.1039/b206378f

M3 - Article

AN - SCOPUS:0036026270

VL - 2

SP - 2137

EP - 2138

JO - Journal of the Chemical Society. Perkin Transactions 1

JF - Journal of the Chemical Society. Perkin Transactions 1

SN - 1470-4358

IS - 19

ER -

Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis

Abstract

ASJC Scopus subject areas

Access to Document

Other files and links

Fingerprint

Cite this