Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis

Kazuo Yamazaki; Yosuke Nakamura; Yoshinori Kondo

doi:10.1039/b206378f

Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis

Kazuo Yamazaki, Yosuke Nakamura, Yoshinori Kondo

PHA - Molecular Pharmaceutical Science

Research output: Contribution to journal › Article › peer-review

43 Citations (Scopus)

Abstract

Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.

Original language	English
Pages (from-to)	2137-2138
Number of pages	2
Journal	Journal of the Chemical Society. Perkin Transactions 1
Volume	2
Issue number	19
DOIs	https://doi.org/10.1039/b206378f
Publication status	Published - 2002 Jul 2

ASJC Scopus subject areas

Chemistry(all)

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abstract = "Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.",

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AU - Nakamura, Yosuke

AU - Kondo, Yoshinori

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N2 - Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.

AB - Intramolecular palladium-catalyzed N-arylation of immobilized dehydrohalophenylalaninate was found to proceed smoothly to form indolecarboxylates. The method was successfully combined with the Heck reaction to perform one pot indole synthesis via palladium-catalyzed tandem C, N-arylation reactions.

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JO - Journal of the Chemical Society. Perkin Transactions 1

JF - Journal of the Chemical Society. Perkin Transactions 1

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ER -

Palladium-catalyzed tandem C, N-arylation of immobilized enamine for solid phase indole synthesis

Abstract

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