Abstract
(Chemical Equation Presented) Catalytic synthesis of 2-substituted benzothiazoles from thiobenzanilides was achieved in the presence of a palladium catalyst through C-H functionalization/C-S bond formation. This method features the use of a novel catalytic system consisting of 10 mol % of Pd(II), 50 mol % of Cu(I), and 2 equiv of Bu4NBr that produced variously substituted benzothiazoles in high yields with good functional group tolerance.
Original language | English |
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Pages (from-to) | 5147-5150 |
Number of pages | 4 |
Journal | Organic letters |
Volume | 10 |
Issue number | 22 |
DOIs | |
Publication status | Published - 2008 Dec 1 |
ASJC Scopus subject areas
- Biochemistry
- Physical and Theoretical Chemistry
- Organic Chemistry