@article{c26ed37fc00e4af3a5792750caae8ece,
title = "Palladium-Catalyzed Highly Chemoselective Intramolecular C-H Aminocarbonylation of Phenethylamines to Six-Membered Benzolactams",
abstract = "A palladium-catalyzed highly selective intramolecular C-H aminocarbonylation of Br-functionalized phenethylamines in the presence of CO was achieved while leaving the C-Br bond unreacted to afford six-membered benzolactams with good to high yields. The remaining C-Br group in the cyclized product was successfully used as a reactive center for further functionalization through various palladium-catalyzed coupling reactions.",
author = "Hiroshi Taneda and Kiyofumi Inamoto and Yoshinori Kondo",
note = "Funding Information: We gratefully acknowledge financial support by a Grant-in-Aid for Scientific Research (B) (No. 23390002), a Grant-in-Aid for Challenging Exploratory Research (No. 25670002), and a Grant-in-Aid for Scientific Research (C) (No. 25460002) from Japan Society for the Promotion of Science, a Grant-in-Aid for Scientific Research on Innovative Areas Advanced Molecular Transformations by Organocatalysis (No. 23105009) and the project Platform for Drug Discovery, Informatics, and Structural Life Science from the Ministry of Education, Culture, Sports, Science and Technology, Japan. Publisher Copyright: {\textcopyright} 2016 American Chemical Society.",
year = "2016",
month = jun,
day = "3",
doi = "10.1021/acs.orglett.6b01171",
language = "English",
volume = "18",
pages = "2712--2715",
journal = "Organic Letters",
issn = "1523-7060",
publisher = "American Chemical Society",
number = "11",
}