3-Methyleneindoline derivatives were synthesized by intramolecular Heck reaction of N-allyl-2-iodoaniline derivatives in the presence of Ag 2CO3. This method was successfully applied to the synthesis of the CC-1065/duocarmycin pharmacophore.
|Number of pages||2|
|Journal||Journal of the Chemical Society, Perkin Transactions 1|
|Publication status||Published - 1993 Jan 1|
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