Abstract
(Chemical Equation Presented) An enantiocontrolled synthesis of (+)-AG-041R (1), a potent gastrin/CCK-B receptor antagonist, has been achieved employing a chiral rhodium(II)-catalyzed, oxidative intramolecular aza-spiroannulation as the key step.
Original language | English |
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Pages (from-to) | 7522-7524 |
Number of pages | 3 |
Journal | Journal of Organic Chemistry |
Volume | 74 |
Issue number | 19 |
DOIs | |
Publication status | Published - 2009 Oct 2 |
ASJC Scopus subject areas
- Organic Chemistry