A new approach to 3-substituted indoles through palladium-catalyzed C-H activation followed by intramolecular amination reaction of enamines

Kiyofumi Inamoto, Tadataka Saito, Kou Hiroya, Takayuki Doi

Research output: Contribution to journalArticle

50 Citations (Scopus)

Abstract

Palladium-catalyzed C-H activation followed by intramolecular amination reaction of enamine compounds was achieved using a Pd(OAc)2 (10 mol%)/Cu(OAc)2 (100 mol%) catalyst system in DMSO. This work introduces an entirely new approach to 3-substituted indoles.

Original languageEnglish
Pages (from-to)3157-3162
Number of pages6
JournalSynlett
Issue number20
DOIs
Publication statusPublished - 2008 Dec 16

Keywords

  • Animations
  • C-H activation
  • Catalysis
  • Indoles
  • Palladium

ASJC Scopus subject areas

  • Organic Chemistry

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